nafarelin  - Drug Details
📊 Estimates nafarelin  Dialyzability By Different_Modalities

nafarelin 

Complete Drug Information

Drug Name
nafarelin 
Trade Names
Synarel, Nasanyl
Bioavailability
INTooltip Intranasal administration: 2.8% (1.2–5.6%)
Routes of Administration
Nasal spray
Protein Binding
80%%
Metabolism
Peptidases (not CYP450Tooltip cytochrome P450)
Elimination
IN: 2.5–3.0 hoursSCTooltip Subcutaneous injection: 86 hours (metabolites)
Excretion
Urine: 44–55%Feces: 19–44%
Formula
C66H83N17O13
Molar Mass
1322.496
Drug Class
GnRH analogue; GnRH agonist; Antigonadotropin
Volume of Distribution
C66H83N17O13