guanfacine  - Drug Details
📊 Estimates guanfacine  Dialyzability By Different_Modalities

guanfacine 

Complete Drug Information

Drug Name
guanfacine 
Trade Names
Intuniv
Bioavailability
80–100% (IR), 58% (XR)
Routes of Administration
Oral
Protein Binding
70%%
Metabolism
CYP3A4
Elimination
IR: 10–17 hours; XR: 17 hours (10–30) in adults & adolescents and 14 hours in children
Excretion
Kidney (80%; 50% [range: 40–75%] as unchanged drug)
Formula
C9H9Cl2N3O
Molar Mass
246.09
Drug Class
α2A-adrenergic receptor agonist
Volume of Distribution
C9H9Cl2N3O