Gabitril - Drug Details
๐Ÿ“Š Estimates Gabitril Dialyzability By Different_Modalities

Gabitril

Complete Drug Information

Drug Name
Gabitril
Trade Names
Gabitril
Bioavailability
90%
Routes of Administration
Oral
Protein Binding
96%%
Metabolism
CYP3A4, possibly other CYP450 enzymes, glucuronidation
Elimination
4.5โ€“9.0 hoursEnzyme-induced patients: 2โ€“3 hours
Excretion
Feces: 63%Urine: 25% (<3% unchanged)
Formula
C20H25NO2S2
Molar Mass
375.55
Onset of Action
1โ€“1.5ย hours
Drug Class
GABA reuptake inhibitor; GABA transporter 1 (GAT-1) inhibitor; Anticonvulsant; Hypnotic; Anxiolytic
Volume of Distribution
C20H25NO2S2