elagolix  - Drug Details
📊 Estimates elagolix  Dialyzability By Different_Modalities

elagolix 

Complete Drug Information

Drug Name
elagolix 
Trade Names
Orilissa, Oriahnn
Pregnancy Category
Contraindicated
Bioavailability
Low (5.8% in rats, 11% in monkeys; no human data)
Routes of Administration
Oral
Protein Binding
80%%
Metabolism
Liver (CYP3A)
Elimination
Typical: 4–6 hoursSingle dose: 2.4–6.3 hrsContinuous: 2.2–10.8 hours
Excretion
Urine: <3%Feces: 90%
Formula
C32H30F5N3O5
Molar Mass
631.6
Drug Class
GnRH antagonist
Volume of Distribution
C32H30F5N3O5

🤰 Pregnancy Category Information

Category: Contraindicated

Pregnancy category: Contraindicated. Consult your healthcare provider for more information.