Zytram - Drug Details
📊 Estimates Zytram Dialyzability By Different_Modalities

Zytram

Complete Drug Information

Drug Name
Zytram
Trade Names
Tramal
Pregnancy Category
AU: C
Bioavailability
68% (by mouth), 77% (rectal), 100% (IM)
Routes of Administration
Oral, intravenous, intramuscular, rectal
Protein Binding
20%%
Metabolism
Liver-mediated demethylation and glucuronidation via CYP2D6 & CYP3A4
Elimination
6.3 ± 1.4 h
Excretion
Urine (95%)
Formula
C16H25NO2
Molar Mass
263.381
Onset of Action
< 1 hour
Duration of Action
6 hours
Melting Point
180 to 181 °C
Drug Class
Opioid; Serotonin–norepinephrine reuptake inhibitor
Volume of Distribution
C16H25NO2

🤰 Pregnancy Category Information

Category: AU: C

Drugs which, owing to their pharmacological effects, have caused or may be suspected of causing harmful effects on the human fetus or neonate without causing malformations. These effects may be reversible.