Zytiga - Drug Details
๐Ÿ“Š Estimates Zytiga Dialyzability By Different_Modalities

Zytiga

Complete Drug Information

Drug Name
Zytiga
Trade Names
Zytiga, Yonsa
Pregnancy Category
AU: D
Bioavailability
Unknown, but may be 50% at most on empty stomach
Routes of Administration
Oral
Protein Binding
Abiraterone: ~99.8% (to albumin and ฮฑ1-AGpTooltip alpha-1 acid glycoprotein)%
Metabolism
Esterases, CYP3A4, SULT2A1
Elimination
Abiraterone: 12โ€“24 hours
Excretion
Feces: 88%Urine: 5%
Formula
C26H33NO2
Molar Mass
391.555
Melting Point
144 to 145ย ยฐC
Drug Class
Antineoplastic
Volume of Distribution
C26H33NO2

๐Ÿคฐ Pregnancy Category Information

Category: AU: D

Drugs which have caused, are suspected to have caused, or may be expected to cause an increased incidence of human fetal malformations or irreversible damage. These drugs may also have adverse pharmacological effects.