Vivitrol - Drug Details
📊 Estimates Vivitrol Dialyzability By Different_Modalities

Vivitrol

Complete Drug Information

Drug Name
Vivitrol
Trade Names
Revia, Vivitrol, Depade
Pregnancy Category
AU: B3
Bioavailability
5–60%
Routes of Administration
Oral, intramuscular, subcutaneous implant
Protein Binding
20%%
Metabolism
Liver (non-CYP450)
Elimination
Oral (Revia):• Naltrexone: 4 hours• 6β-Naltrexol: 13 hoursOral (Contrave):• Naltrexone: 5 hoursIMTooltip Intramuscular injection (Vivitrol):• Naltrexone: 5–10 days• 6β-Naltrexol: 5–10 days
Excretion
Urine
Formula
C20H23NO4
Molar Mass
341.407
Onset of Action
30 minutes
Duration of Action
>72 hours
Melting Point
169 °C
Volume of Distribution
C20H23NO4

🤰 Pregnancy Category Information

Category: AU: B3

Drugs which have been taken by only a limited number of pregnant women and women of childbearing age, without an increase in the frequency of malformation or other direct or indirect harmful effects on the human fetus. Animal studies have shown evidence of an increased occurrence of fetal damage, the significance of which is considered uncertain in humans.