efavirenz  - Drug Details
📊 Estimates efavirenz  Dialyzability By Different_Modalities

efavirenz 

Complete Drug Information

Drug Name
efavirenz 
Trade Names
Sustiva, Stocrin
Pregnancy Category
AU: D
Bioavailability
40–45% (under fasting conditions)
Routes of Administration
Oral (capsules, tablets)
Protein Binding
99.5–99.75%%
Metabolism
Liver (CYP2A6 and CYP2B6-mediated)
Elimination
Single-dose: 52–76 hMulti-dose: 40–55 h
Excretion
Kidney (14–34%) and feces (16–61%)
Formula
C14H9ClF3NO2
Molar Mass
315.68
Onset of Action
3–5 hours
Volume of Distribution
2 L/kg

🤰 Pregnancy Category Information

Category: AU: D

Drugs which have caused, are suspected to have caused, or may be expected to cause an increased incidence of human fetal malformations or irreversible damage. These drugs may also have adverse pharmacological effects.