varenicline - Drug Details
๐Ÿ“Š Estimates varenicline Dialyzability By Different_Modalities

varenicline

Complete Drug Information

Drug Name
varenicline
Trade Names
Champix, Chantix, Tyrvaya
Pregnancy Category
AU: B3
Routes of Administration
Oral, intranasal
Protein Binding
<20%%
Metabolism
Primarily unchanged by OCT2. Insignificant CYP450 enzyme involved
Elimination
24 hours
Excretion
Kidney (81โ€“92%)
Formula
C13H13N3
Molar Mass
211.268
Drug Class
Nicotinic agonist
Volume of Distribution
415 L/kg

๐Ÿคฐ Pregnancy Category Information

Category: AU: B3

Drugs which have been taken by only a limited number of pregnant women and women of childbearing age, without an increase in the frequency of malformation or other direct or indirect harmful effects on the human fetus. Animal studies have shown evidence of an increased occurrence of fetal damage, the significance of which is considered uncertain in humans.