mexiletine  - Drug Details
📊 Estimates mexiletine  Dialyzability By Different_Modalities

mexiletine 

Complete Drug Information

Drug Name
mexiletine 
Trade Names
Mexitil, NaMuscla
Pregnancy Category
AU: B1
Bioavailability
90%
Routes of Administration
Oral, intravenous
Protein Binding
50–60%%
Metabolism
Liver (CYP2D6 and 1A2-mediated)
Elimination
10–12 hours
Excretion
Kidney (10%)
Formula
C11H17NO
Molar Mass
179.263
Volume of Distribution
5 L/kg

🤰 Pregnancy Category Information

Category: AU: B1

Drugs which have been taken by only a limited number of pregnant women and women of childbearing age, without an increase in the frequency of malformation or other direct or indirect harmful effects on the human fetus. Animal studies have not shown evidence of an increased occurrence of fetal damage.