macitentan  - Drug Details
📊 Estimates macitentan  Dialyzability By Different_Modalities

macitentan 

Complete Drug Information

Drug Name
macitentan 
Trade Names
Opsumit
Pregnancy Category
AU: X (High risk)
Routes of Administration
Oral
Metabolism
Hydrolysis, oxidation (CYP3A4)
Excretion
2/3 urine, 1/3 faeces
Formula
C19H20Br2N6O4S
Molar Mass
588.28
Volume of Distribution
50 L/kg

🤰 Pregnancy Category Information

Category: AU: X (High risk)

Drugs which have such a high risk of causing permanent damage to the fetus that they should not be used in pregnancy or when there is a possibility of pregnancy.