lofepramine  - Drug Details
📊 Estimates lofepramine  Dialyzability By Different_Modalities

lofepramine 

Complete Drug Information

Drug Name
lofepramine 
Trade Names
Gamanil, Lomont, Tymelyt
Bioavailability
7%
Routes of Administration
Oral
Protein Binding
99%%
Metabolism
Hepatic (via cytochrome P450, including CYP2D6)
Elimination
Up to 5 hours; 12–24 hours (active metabolites)
Excretion
Urine, feces (mostly as metabolites)
Formula
C26H27ClN2O
Molar Mass
418.97
Volume of Distribution
C26H27ClN2O