leflunomide  - Drug Details
📊 Estimates leflunomide  Dialyzability By Different_Modalities

leflunomide 

Complete Drug Information

Drug Name
leflunomide 
Trade Names
Arava, Lefumide, Arabloc
Pregnancy Category
AU: X (High risk)
Bioavailability
80%
Routes of Administration
Oral
Protein Binding
>99%%
Metabolism
GI mucosa and liver
Elimination
14–18 days
Excretion
Faeces (48%), urine (43%)
Formula
C12H9F3N2O2
Molar Mass
270.211
Volume of Distribution
11 L/kg

🤰 Pregnancy Category Information

Category: AU: X (High risk)

Drugs which have such a high risk of causing permanent damage to the fetus that they should not be used in pregnancy or when there is a possibility of pregnancy.