lapatinib_ditosylate  - Drug Details
📊 Estimates lapatinib_ditosylate  Dialyzability By Different_Modalities

lapatinib_ditosylate 

Complete Drug Information

Drug Name
lapatinib_ditosylate 
Trade Names
Tykerb, Tyverb
Pregnancy Category
AU: C
Bioavailability
Variable, increased with food
Routes of Administration
Oral
Protein Binding
>99%%
Metabolism
Liver, mostly CYP3A-mediated (minor 2C19 and 2C8 involvement)
Elimination
24 hours (repeated dosing), 14.2 hours (single dose)
Excretion
Mostly Feces
Formula
C29H26ClFN4O4S
Molar Mass
581.06
Volume of Distribution
C29H26ClFN4O4S

🤰 Pregnancy Category Information

Category: AU: C

Drugs which, owing to their pharmacological effects, have caused or may be suspected of causing harmful effects on the human fetus or neonate without causing malformations. These effects may be reversible.