labetalol  - Drug Details
📊 Estimates labetalol  Dialyzability By Different_Modalities

labetalol 

Complete Drug Information

Drug Name
labetalol 
Trade Names
Normodyne, Trandate
Pregnancy Category
AU: C
Bioavailability
25% (11–86%)
Routes of Administration
Oral, intravenous
Protein Binding
50%%
Metabolism
Mainly conjugation via glucuronidation
Elimination
Oral: 6–8 hoursIVTooltip Intravenous infusion: 5.52 hours
Excretion
Urine (55–60% as conjugates or unchanged within 24 hours)
Formula
C19H24N2O3
Molar Mass
328.412
Duration of Action
8–12 hours
Volume of Distribution
5.6 L/kg

🤰 Pregnancy Category Information

Category: AU: C

Drugs which, owing to their pharmacological effects, have caused or may be suspected of causing harmful effects on the human fetus or neonate without causing malformations. These effects may be reversible.