Oleptro - Drug Details
📊 Estimates Oleptro Dialyzability By Different_Modalities

Oleptro

Complete Drug Information

Drug Name
Oleptro
Trade Names
Desyrel, Trittico
Bioavailability
By mouth: 63–80%
Routes of Administration
Oral
Protein Binding
89–95%%
Metabolism
Liver (CYP3A4, CYP2D6, CYP1A2?)
Elimination
• Trazodone (IR): 4–15 hours• Trazodone (ER): 9–13 hours• mCPPTooltip meta-Chlorophenylpiperazine: 3–16 hours
Excretion
Urine: 70–75%Feces: 21%
Formula
C19H22ClN5O
Molar Mass
371.87
Onset of Action
1 hour
Melting Point
87 °C
Drug Class
Serotonin antagonist and reuptake inhibitor (SARI); Serotonin 5-HT2A receptor antagonist; α1-Adrenergic receptor antagonist; Serotonin reuptake inhibitor
Volume of Distribution
C19H22ClN5O