olanzapine  - Drug Details
📊 Estimates olanzapine  Dialyzability By Different_Modalities

olanzapine 

Complete Drug Information

Drug Name
olanzapine 
Trade Names
Zyprexa
Pregnancy Category
AU: C
Bioavailability
60–65%
Routes of Administration
Oral, intramuscular
Protein Binding
93%%
Metabolism
Liver (direct glucuronidation and CYP1A2 mediated oxidation)
Elimination
33 hours, 51.8 hours (elderly)
Excretion
Urine (57%; 7% as unchanged drug), faeces (30%)
Formula
C17H20N4S
Molar Mass
312.44
Melting Point
195 °C
Drug Class
Atypical antipsychotic
Volume of Distribution
10 L/kg

🤰 Pregnancy Category Information

Category: AU: C

Drugs which, owing to their pharmacological effects, have caused or may be suspected of causing harmful effects on the human fetus or neonate without causing malformations. These effects may be reversible.